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VORAXAZE® (glucarpidase) Mechanism of Action for Methotrexate Toxicity Secondary to Renal Impairment
Daim Duab: VORAXAZE® (glucarpidase) Mechanism of Action for Methotrexate Toxicity Secondary to Renal Impairment

Zoo Siab

Glucarpidase yog siv los tiv thaiv kev puas tsuaj ntawm methotrexate (Rheumatrex, Trexall) rau cov neeg mob raum uas tau txais methotrexate los kho qee yam mob qog ntshav. Glucarpidase yog nyob hauv chav kawm ntawm cov tshuaj hu ua enzymes. Nws ua haujlwm los ntawm kev pab rhuav tshem thiab tshem methotrexate tawm ntawm lub cev.

Glucarpidase los ua hmoov los tov nrog kua thiab txhaj koob txhaj tshuaj (rau hauv cov leeg ntshav). Nws ib txwm muab li 5 feeb ua ib zaug. Glucarpidase tau muab nrog leucovorin (lwm cov tshuaj siv los tiv thaiv kev puas tsuaj ntawm methotrexate) txog thaum kuaj sim pom tias yuav kho tsis tau ntxiv lawm.

Cov tshuaj no tuaj yeem tsim tawm rau lwm txoj kev siv; nug koj tus kws kho mob lossis kws muag tshuaj kom paub ntaub ntawv ntau ntxiv.

Ua ntej noj glucarpidase,

  • qhia rau koj tus kws kho mob thiab kws muag tshuaj yog tias koj muaj kev fab tshuaj rau glucarpidase, lwm yam tshuaj noj, lossis ib qho twg ntawm cov khoom xyaw txhaj tshuaj glucarpidase. Nug koj tus kws muag tshuaj rau cov npe ntawm cov khoom xyaw.
  • qhia rau koj tus kws kho mob thiab kws muag tshuaj tias lwm yam tshuaj uas tsis yog kws kho mob thiab cov tshuaj uas tsis yog kws kho mob sau, tshuaj vitamins, khoom noj khoom haus zoo, thiab tshuaj ntsuab koj tau noj lossis npaj yuav noj. Nco ntsoov hais txhua yam ntawm cov hauv qab no: folic acid (Folicet, hauv multivitamins); levoleucovorin (Fusilev); lossis pemetrexed (Alimta). Koj tus kws kho mob tej zaum yuav tau hloov qhov tshuaj ntawm koj cov tshuaj lossis saib xyuas koj kom zoo rau kev phiv.
  • yog tias koj tau txais leucovorin, nws yuav tsum muab tsawg kawg 2 teev ua ntej lossis 2 teev tom qab glucarpidase.
  • qhia koj tus kws kho mob yog tias koj cev xeeb tub, npaj yuav cev xeeb tub, lossis pub mis niam. Yog tias koj xeeb tub thaum noj cov tshuaj glucarpidase, hu rau koj tus kws kho mob.

Tshwj tsis yog koj tus kws kho mob hais rau koj lwm yam, txuas ntxiv koj li kev noj haus zoo.


Glucarpidase tuaj yeem tshwm sim phiv. Qhia rau koj tus kws kho mob yog tias ib qho ntawm cov tsos mob no hnyav lossis tsis ploj mus:

  • xeev siab
  • ntuav

Qee qhov kev mob tshwm sim tuaj yeem loj heev. Yog tias koj muaj cov tsos mob no, hu rau koj tus kws kho mob sai lossis tau txais kev kho mob kub ceev:

  • ua npaws
  • ua daus no
  • plhu lossis hnov ​​kub
  • ua pob
  • khaus
  • khaus
  • caj pas nruj los yog ua pa nyuaj
  • cov kev xav ntawm loog, tingling, pricking, hlawv, lossis hma ntawm daim tawv nqaij
  • mob taub hau

Glucarpidase tuaj yeem ua lwm cov kev mob tshwm sim. Hu rau koj tus kws kho mob yog tias koj muaj teeb meem txawv txawv thaum noj cov tshuaj no.

Yog tias koj muaj kev mob tshwm sim loj, koj lossis koj tus kws kho mob tuaj yeem xa ntawv ceeb toom rau Food and Drug Administration's (FDA) MedWatch Adverse Event Reporting program online (http://www.fda.gov/Safety/MedWatch) lossis hauv xov tooj ( 1-800-332-1088).

Khaws tag nrho cov kev teem caij mus ntsib koj tus kws kho mob thiab chav kuaj mob. Koj tus kws kho mob yuav xaj qee yam kev kuaj sim kuaj xyuas koj lub cev cov lus teb rau glucarpidase.


Nug koj tus kws muag tshuaj yog tias koj muaj lus nug dab tsi txog glucarpidase.

Nws yog ib qho tseem ceeb rau koj kom koj muaj ib daim ntawv sau tag nrho cov tshuaj noj thiab cov tshuaj uas tsis yog kws kho mob sau ntawv (tsis yuav khoom) uas koj tab tom noj, nrog rau txhua yam khoom xws li cov vitamins, minerals, lossis lwm yam tshuaj noj rau lub cev. Koj yuav tsum nqa cov ntawv no nrog koj txhua zaus koj mus ntsib kws kho mob lossis yog tias koj tuaj nyob hauv tsev kho mob. Nws tseem yog cov ntaub ntawv tseem ceeb los nqa nrog koj thaum muaj xwm txheej ceev.

  • Voraxaze®
Kawg Siv - 02/15/2013

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